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Improvement in oral bioavailability of 2,4-diaminopyrimidine c-Met inhibitors by incorporation of a 3-amidobenzazepin-2-one group

作者:Karen L. Milkiewicz, Lisa D. Aimone, Mark S. Albom, Thelma S. Angeles, Hong Chang, Jennifer V. Grobelny, Jean Husten, Christine LoSardo, Sheila Miknyoczki, S. N. Prasanna Murthy, Damaris Rolon-Steele, Ted L. Underiner, Linda R. Weinberg, Candace S. Worrell, Kelli S. Zeigler, Bruce D. Dorsey · 发表于:Bioorganic & Medicinal Chemistry · 年份:2011 · DOI:10.1016/j.bmc.2011.09.006 · 被引用次数:14 · 研究领域:Liver physiology and pathology、Hepatocellular Carcinoma Treatment and Prognosis、Drug-Induced Hepatotoxicity and Protection