Discovery of a brain-permeable bromodomain and extra terminal domain (BET) inhibitor with selectivity for BD1 for the treatment of multiple sclerosis
作者:Xuetao Chen, Tingting Wu, Zhiyan Du, Wenjing Kang, Rujun Xu, Fanying Meng, Chihong Liu, Yali Chen, Qichao Bao, Jingkang Shen, Qidong You, Danyan Cao, Zhengyu Jiang, Xiaoke Guo · 发表于:European Journal of Medicinal Chemistry · 年份:2023 · DOI:10.1016/j.ejmech.2023.116080 · 被引用次数:14 · 研究领域:Protein Degradation and Inhibitors、Multiple Myeloma Research and Treatments、RNA Interference and Gene Delivery