Azaindole N-methyl hydroxamic acids as HIV-1 integrase inhibitors-II. The impact of physicochemical properties on ADME and PK
作者:Steven P. Tanis, Michael Plewe, Ted W. Johnson, Scott L. Butler, Deepak Dalvie, Dorothy M. DeLisle, Klaus Dress, Qiyue Hu, Buwen Huang, Jon Kuehler, Atsuo Kuki, Wen Liu, Qinghai Peng, Graham L. Smith, Jim Solowiej, Khanh Tran, Hai Wang, Anle Yang, Chunfeng Yin, Xiaoming Yu, Junhu Zhang, Huichun Zhu · 发表于:Bioorganic & Medicinal Chemistry Letters · 年份:2010 · DOI:10.1016/j.bmcl.2010.10.022 · 被引用次数:23 · 研究领域:HIV/AIDS drug development and treatment、HIV Research and Treatment、Pneumocystis jirovecii pneumonia detection and treatment