Design, synthesis, and biological evaluation of N-(2-amino-phenyl)-5-(4-aryl- pyrimidin-2-yl) amino)-1H-indole-2-carboxamide derivatives as novel inhibitors of CDK9 and class I HDACs for cancer treatment
作者:Xiaohui Chen, Rongna Li, Ying‐Kun Qiu, F. Lin, Shutong Chen, Xiaodan Li, Hui Sun, Guanmin Jiang, Hua Fang, Jingbo Qin, Meijuan Fang · 发表于:Bioorganic Chemistry · 年份:2025 · DOI:10.1016/j.bioorg.2025.108577 · 被引用次数:8 · 研究领域:Histone Deacetylase Inhibitors Research、Peptidase Inhibition and Analysis、Click Chemistry and Applications