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Design, synthesis, anti-tumor activity and mechanism of novel PROTACs as degraders of PD-L1 and inhibitors of PD-1/PD-L1 interaction

作者:Feng Zhang, Feng Zhang, Caiyun Wu, Caiyun Wu, Shishi Sun, Yu Wang, Rui Wang, Zejie Chen, Hua Zhang, Hua Zhang, Xuqiong Xiong, Annoor Awadasseid, Guo‐Wu Rao, Xiaoyin Zhao, Wen Zhang · 发表于:Bioorganic & Medicinal Chemistry · 年份:2024 · DOI:10.1016/j.bmc.2024.117867 · 被引用次数:13 · 研究领域:Protein Degradation and Inhibitors、CAR-T cell therapy research、Peptidase Inhibition and Analysis