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Discovery and characterization of novel potent BCR-ABL degraders by conjugating allosteric inhibitor

作者:Haixia Liu, Qianglong Mi, Xinyu Ding, Chencen Lin, Linyi Liu, Chaowei Ren, ShuTing Shen, Yubao Shao, Jinju Chen, Yongqi Zhou, Liting Ji, Heqiao Zhang, Fang Bai, Xiaobao Yang, Qianqian Yin, Biao Jiang · 发表于:European Journal of Medicinal Chemistry · 年份:2022 · DOI:10.1016/j.ejmech.2022.114810 · 被引用次数:31 · 研究领域:Protein Degradation and Inhibitors、Multiple Myeloma Research and Treatments、Peptidase Inhibition and Analysis