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Design, synthesis and biological evaluation of potent EGFR kinase inhibitors against 19D/T790M/C797S mutation

作者:Zhicheng Su, Tingyuan Yang, Jie Wang, Mengzhen Lai, Linjiang Tong, Gulinuer Wumaier, Zhuo Chen, Shengqing Li, Honglin Li, Hua Xie, Zhenjiang Zhao · 发表于:Bioorganic & Medicinal Chemistry Letters · 年份:2020 · DOI:10.1016/j.bmcl.2020.127327 · 被引用次数:24 · 研究领域:Lung Cancer Treatments and Mutations、Cancer therapeutics and mechanisms、HER2/EGFR in Cancer Research