Discovery of a series of dihydroquinoxalin-2(1H)-ones as selective BET inhibitors from a dual PLK1-BRD4 inhibitor

作者：Jianping Hu, Ying-Qing Wang, Yanlian Li, Lin Xu, Danyan Cao, Shanshan Song, Mohammadali Soleimani Damaneh, Xin Wang, Tao Meng, Yue‐Lei Chen, Jingkang Shen, Ze‐Hong Miao, Bing Xiong · 发表于：European Journal of Medicinal Chemistry · 年份：2017 · DOI：10.1016/j.ejmech.2017.05.049 · 被引用次数：36 · 研究领域：Protein Degradation and Inhibitors、Multiple Myeloma Research and Treatments、Ubiquitin and proteasome pathways