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Bioavailable pyrrolo-benzo-1,4-diazines as Nav1.7 sodium channel blockers for the treatment of pain

作者:Shu‐Wei Yang, Ginny D. Ho, Deen Tulshian, Ana Bercovici, Zheng Tan, Jennifer Hanisak, Stephanie Brumfield, Julius J. Matasi, Xianfeng Sun, Samuel A. Sakwa, R. Jason Herr, Xiaoping Zhou, Terry Bridal, Mark O. Urban, Jeffrey A. Vivian, Diane Rindgen, Steve Sorota · 发表于:Bioorganic & Medicinal Chemistry Letters · 年份:2014 · DOI:10.1016/j.bmcl.2014.09.038 · 被引用次数:15 · 研究领域:Ion channel regulation and function、Pain Mechanisms and Treatments、Synthesis and Reactivity of Heterocycles