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Identification of amides derived from 1H-pyrazolo[3,4-b]pyridine-5-carboxylic acid as potent inhibitors of human nicotinamide phosphoribosyltransferase (NAMPT)

作者:Xiaozhang Zheng, Kenneth W. Bair, Paul Bauer, Timm Baumeister, Krista K. Bowman, Alexandre J. Buckmelter, Maureen Caligiuri, Karl H. Clodfelter, Y. Feng, Bingsong Han, Yen‐Ching Ho, Nikolai Kley, Hong Li, Xiaorong Liang, Bianca M. Liederer, Jian Lin, Justin Q. Ly, Thomas O’Brien, Jason Oeh, Angela Oh, Dominic J. Reynolds, Deepak Sampath, Geeta Sharma, Nicholas J. Skelton, Chase C. Smith, Jarrod R. Tremayne, Leslie Wang, Weiru Wang, Zhongguo Wang, Hongxing Wu, Jiansheng Wu, Yang Xiao, Guangxing Yang, Po‐wai Yuen, Mark Zak, Peter S. Dragovich · 发表于:Bioorganic & Medicinal Chemistry Letters · 年份:2013 · DOI:10.1016/j.bmcl.2013.08.074 · 被引用次数:45 · 研究领域:Calcium signaling and nucleotide metabolism、Biochemical and Molecular Research、Sirtuins and Resveratrol in Medicine