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Rita L. Civiello

机构:Bristol-Myers Squibb (Germany), Bristol-Myers Squibb (Belgium)

发表论文 35 篇 · 总被引 779 次 · h-index 14

代表论文

  • Discovery of new acylaminopyridines as GSK-3 inhibitors by a structure guided in-depth exploration of chemical space around a pyrrolopyridinone core (2015 · Bioorganic & Medicinal Chemistry Letters · 被引 117)
  • Respiratory syncytial virus fusion inhibitors. Part 7: Structure–activity relationships associated with a series of isatin oximes that demonstrate antiviral activity in vivo (2009 · Bioorganic & Medicinal Chemistry Letters · 被引 46)
  • Respiratory syncytial virus fusion inhibitors. Part 6: An examination of the effect of structural variation of the benzimidazol-2-one heterocycle moiety (2007 · Bioorganic & Medicinal Chemistry Letters · 被引 40)
  • Respiratory syncytial virus fusion inhibitors. Part 5: Optimization of benzimidazole substitution patterns towards derivatives with improved activity (2007 · Bioorganic & Medicinal Chemistry Letters · 被引 33)
  • Syntheses of aza and fluorine-substituted 3-(piperidin-4-yl)-4,5-dihydro-1H-benzo[d][1,3]diazepin-2(3H)-ones (2008 · Tetrahedron Letters · 被引 26)
  • Calcitonin gene-related peptide (CGRP) receptor antagonists: Pyridine as a replacement for a core amide group (2012 · Bioorganic & Medicinal Chemistry Letters · 被引 21)