Patrick R. Gentry

机构：Australian Regenerative Medicine Institute, Monash University · ORCID：0000-0003-0670-6648

发表论文 58 篇 · 总被引 2080 次 · h-index 23

代表论文

• Novel Allosteric Modulators of G Protein-coupled Receptors (2015 · Journal of Biological Chemistry · 被引 203)
• Crystal structure of the M 5 muscarinic acetylcholine receptor (2019 · Proceedings of the National Academy of Sciences · 被引 84)
• Discovery of ( S )-2-Cyclopentyl- N -((1-isopropylpyrrolidin2-yl)-9-methyl-1-oxo-2,9-dihydro-1 H -pyrrido[3,4- b ]indole-4-carboxamide (VU0453379): A Novel, CNS Penetrant Glucagon-Like Peptide 1 Receptor (GLP-1R) Positive Allosteric Modulator (PAM) (2014 · Journal of Medicinal Chemistry · 被引 47)
• Molecular insights into ligand recognition and G protein coupling of the neuromodulatory orphan receptor GPR139 (2021 · Cell Research · 被引 37)
• Discovery, Synthesis and Characterization of a Highly Muscarinic Acetylcholine Receptor (mAChR)‐Selective M 5 ‐Orthosteric Antagonist, VU0488130 (ML381): A Novel Molecular Probe (2014 · ChemMedChem · 被引 34)
• Molecular Mechanisms of Action of M5 Muscarinic Acetylcholine Receptor Allosteric Modulators (2016 · Molecular Pharmacology · 被引 33)