Peter H. Crackett

机构：Charles River Laboratories (United Kingdom)

发表论文 34 篇 · 总被引 557 次 · h-index 12

代表论文

• Studies toward the Large-Scale Synthesis of the HIV Proteinase Inhibitor Ro 31-8959 (1994 · The Journal of Organic Chemistry · 被引 98)
• Identification of C-2 Hydroxyethyl Imidazopyrrolopyridines as Potent JAK1 Inhibitors with Favorable Physicochemical Properties and High Selectivity over JAK2 (2013 · Journal of Medicinal Chemistry · 被引 63)
• Discovery of a class of highly potent Janus Kinase 1/2 (JAK1/2) inhibitors demonstrating effective cell-based blockade of IL-13 signaling (2019 · Bioorganic & Medicinal Chemistry Letters · 被引 59)
• 1H-Pyrazolo[3,4-g]hexahydro-isoquinolines as selective glucocorticoid receptor antagonists with high functional activity (2008 · Bioorganic & Medicinal Chemistry Letters · 被引 50)
• Asymmetric synthesis via acetal templates. 9. Further studies of the allylation reaction. Preparation of (−)-dihydromyoporone (1984 · Tetrahedron Letters · 被引 50)
• Complexes of imidazoline (1,3H)-2-thione with Co(II) and Zn(II) salts (1981 · Inorganica Chimica Acta · 被引 41)