David J. Augeri

机构：Rutgers, The State University of New Jersey, Schrodinger (United States)

发表论文 54 篇 · 总被引 5640 次 · h-index 20

代表论文

• An inhibitor of Bcl-2 family proteins induces regression of solid tumours (2005 · Nature · 被引 3429)
• Discovery and Preclinical Profile of Saxagliptin (BMS-477118): A Highly Potent, Long-Acting, Orally Active Dipeptidyl Peptidase IV Inhibitor for the Treatment of Type 2 Diabetes (2005 · Journal of Medicinal Chemistry · 被引 625)
• Discovery of a Potent Inhibitor of the Antiapoptotic Protein Bcl-x L from NMR and Parallel Synthesis (2005 · Journal of Medicinal Chemistry · 被引 297)
• NMR-Based Screening of Proteins Containing 13C-Labeled Methyl Groups (2000 · Journal of the American Chemical Society · 被引 209)
• Novel Inhibitors of Erm Methyltransferases from NMR and Parallel Synthesis (1999 · Journal of Medicinal Chemistry · 被引 121)
• Inhibition of Sphingosine 1-Phosphate Lyase for the Treatment of Rheumatoid Arthritis: Discovery of (E)-1-(4-((1R,2S,3R)-1,2,3,4-Tetrahydroxybutyl)-1H-imidazol-2-yl)ethanone Oxime (LX2931) and (1R,2S,3R)-1-(2-(Isoxazol-3-yl)-1H-imidazol-4-yl)butane-1,2,3,4-tetraol (LX2932) (2010 · Journal of Medicinal Chemistry · 被引 113)